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2019年

作者：  来源：  发布日期：2020年06月09日
  1. Jianzhong Liu, Cheng Zhang, Ziyao Zhang, Xiaojin Wen, Xiaodong Dou, Jialiang Wei, Xu Qiu, Song Song, Ning Jiao*. Nitromethane as a nitrogen donor in Schmidt-type formation of amides and nitriles. Science, 2019, DOI: 10.1126/science.aay9501.
  2. Bencong Zhu, Tao Shen, Xiaoqiang Huang, Yuchao Zhu, Song Song, and Ning Jiao*. Selective Aerobic Oxygenation of Tertiary Allylic Alcohols with Molecular Oxygen. Angew. Chem. Int. Ed., 2019, 58, 11028-11032.
  3. Qixue Qin, Xiao Luo, Jialiang Wei, Yuchao Zhu, Xiaojin Wen, Song Song, and Ning Jiao*. Acetonitrile Activation: An Effective C2 Cyclization Unit. Angew. Chem. Int. Ed., 2019, 58, 4420-4424.
  4. Yujie Liang, Fengguirong Lin, Yeerlan Adeli, Rui Jin, and Ning Jiao*. Efficient electrocatalysis for the preparation of (hetero)aryl chlorides and vinyl chloride with 1,2-dichloroethane. Angew. Chem. Int. Ed., 2019, 58, 4566-4570.
  5. Jianzhong Liu, Xu Qiu, Xiaoqiang Huang, Xiao Luo, Jialiang Wei, Jun Pan, Yujie Liang, Yuchao Zhu, Qixue Qin, Song Song, and Ning Jiao*. From Alkylarenes to Anilines via Site-Directed Carbon-Carbon Amination. Nature Chemistry, 2019, 11, 71-77.
  6. Yeerlan Adeli, Kaimeng Huang, Yujie Liang, Yangye Jiang, Jianzhong Liu, Song Song, Cheng-Chu Zeng* and Ning Jiao*. Electrochemically Oxidative C-C Bond Cleavage of Alkylarenes for Anilines Synthesis. ACS Catal., 2019, 9 (3), 2063-2067.
  7. Junhua Li, Jialiang Wei, Bencong Zhu, Teng Wang, and Ning Jiao*. Cu-catalyzed Oxygenation of Alkene-tethered Amides with O2 via Unactivated C=C Bond Cleavage: A Direct Approach to Cyclic Imides. Chem. Sci., 2019, 10, 9099–9103.
  8. Qixue Qin, Weijing Wang, Cheng Zhang, Song Song*, Ning Jiao*. A metal-free desulfurizing Radical Reductive C-C Coupling of Thiols and Alkenes. Chem. Commun., 2019, 55, 10583-10586.
  9. Lingsheng Ai, Weijin Wang, Jialiang Wei, Qing Li, Song Song*, and Ning Jiao*. Oxidative β-Halogenation of Alcohols: A Concise and Diastereoselective Approach to Halohydrins. Synlett., 2019, 30, 437-441.
  10. Xu Qiu, Xiaoxue Yang, Yiqun Zhang, Song Song*, Ning Jiao. Efficient and Practical Synthesis of Unsymmetrical Disulfides via Base-Catalyzed Aerobic Oxidative Dehydrogenative Coupling of Thiols. Organic Chemistry Frontiers, 2019, 6, 2220-2225.
  11. Yuan Ma, Wenting Zhao, Yiding Li, Yufei Pan, Shuhe Wang, Yuejie Zhu, Lingxuan Kong, Zhu Guan, Jiancheng Wang, Lihe Zhang, Zhenjun Yang*. Structural optimization and additional targets identification of antisense oligonucleotide G3139 encapsulated in a neutral cytidinyl-lipid combined with a cationic lipid in vitro and in vivo. Biomaterials, 2019, 197, 182-193.
  12. Lei Li, Kuo Yuan, Qianlan Jia, Yanxing Jia*. Eight-Step Total Synthesis of Phalarine by Bioinspired Oxidative Coupling of Indole and Phenol. Angew. Chem. Int. Ed., 2019, 58(18), 6074–6078.
  13. Haichao Liu, Lijun Chen, Kuo Yuan, Yanxing Jia*. A Ten-Step Total Synthesis of Speradine C. Angew. Chem. Int. Ed., 2019, 58(19), 6362–6365.
  14. Xiwu Zhang, Xinxian Cai, Bin Huang, Lei Guo, Zhongrun Gao, Yanxing Jia*. Enantioselective Total Syntheses of Pallambins A-D. Angew. Chem. Int. Ed., 2019, 58(38), 13380–13384.
  15. Xiaodong Dou, Huixia Huang, Yibo Li, Lan Jiang, Yanxing Wang, Hongwei Jin, Ning Jiao, Lihe Zhang, Liangren Zhang*, Zhenming Liu*. Multistage Screening Reveals 3-Substituted lndolin-2-one Derivatives as Novel and Isoform-Selective c-Jun N-terminal Kinase 3 (JNK3) Inhibitors: Implications to Drug Discovery for Potential Treatment of Neurodegenerative Diseases. J. Med. Chem., 2019, 62, 6645-6664.
  16. QingQing Jin, Xinli Fan, Changmai Chen, Lei Huang, Jing Wang, Xinjing Tang*. Multicolor Raman Beads for Multiplexed Tumor Cell and Tissue Imaging and in Vivo Tumor Spectral Detection. Anal. Chem., 2019, 91, 3784？3789.
  17. Changmai Chen, Zhongyu Wang, Jinhao Zhang, Xinli Fan, Luzheng Xu, and Xinjing Tang*. Dextran-Conjugated Caged siRNA Nanoparticles for Photochemical Regulation of RNAi-Induced Gene Silencing in Cells and Mice. Bioconjugate Chem., 2019, 30, 5, 1459-1465.
  18. Jie Feng, Jiale Zhong and Xinjing Tang*. Selective and sensitive detection of cyanate using 3-amino-2-naphthoic acid-based turn-on fluorescence probe. Anal. Bioanal. Chem., 2019, 411, 3613–3619.
  19. Jie Feng, Xiaoran Zhao, Wei Bian and Xinjing Tang*. Microwave-assisted synthesis of nitrogen-rich carbon dots as effective fluorescent probe for sensitive detection of Ag+
  20. Materials Chemistry Frontiers, 2019, DOI: 10.1039/C9QM00624A.
  21. Xiling Bian*, Yu Zhang, Bin Huang, Xintong Wang, Gongxin Wang, Yuhao Zhu, Yan Liu, Jianhui Liang, Yanxing Jia*, KeWei Wang*. Natural product incarvillateine aggravates epileptic seizures by inhibiting GABAA currents. Eur. J. Pharmaco. 2019, 858, 172496.
  22. Yang Wang, Kang Liu, Zhi-Xiang Yu*, Yanxing Jia*. Type-II Pauson-Khand Reaction of 1,8-enyne in the Attempt of Building 7/5 Ring of (-)-Caribenol A and DFT Understanding. Tetrahedron. Lett., 2019, 60 (36), 151001.
  23. Dandan Xi, Yan Niu*, Hongyue Li, Stefan M. Noha, Veronika Temml, Daniela Schuster*, Chao Wang, Fengrong Xu, and Ping Xu*. Discovery of carbazole derivatives as novel allosteric MEK inhibitors by pharmacophore modeling and virtual screening. Eur. J. Med. Chem., 2019,178, 802-817.
  24. Hongyue Li, Dandan Xi, Yan Niu, Chao Wang, Fengrong Xu, Lei Liang*, Ping Xu*. Design, synthesis and biological evaluation of cobalt(II)-Schiff base complexes as ATP-noncompetitive MEK1 inhibitors. J. Inorg. Biochem.2019, 195, 174-181.
  25. Xiufeng Xu, Peng Lü, Junjie Wang, Fengrong Xu, Lei Liang, Chao Wang, Yan Niu*, Ping Xu*. Design, synthesis, and biological evaluation of 4-aminopyrimidine or 4,6-diaminopyrimidine derivatives as beta amyloid cleaving enzyme-1 inhibitors. Chem. Biol. Drug. Des. 2019, 93(5), 926-933.
  26. Shuobin Liang, Man Li, Xiaojuan Yu, Hongwei Jin, Yongmin Zhang, Lihe Zhang, Demin Zhou, Sulongxiao*. Synthesis and structure-activity relationship studies of water-soluble β-cyclodextrin-glycyrrhetinic acid conjugates as potential anti-influenza virus agents. Eur. J. Med. Chem., 2019, 166, 328-338.
  27. Haiwei Li, Man Li, Renyang Xu, Shouxin Wang, Yongmin Zhang, Lihe Zhang, Demin Zhou*, Sulong Xiao*. Synthesis, structure activity relationship and in vitro anti-influenza virus activity of novel polyphenol-pentacyclic triterpene conjugates. Eur. J. Med. Chem., 2019, 163, 560-568.
  28. DaKe Liu, DeCai Xiong, Xia Wu, Qin Li*, XinShan Ye*. Rapid glycosylation of 2’-benzoylphenyl glycosides promoted by TfOH. Org. Chem. Frontiers, 2019, 6, 2756–2759.
  29. Yanxing Wang, Xiaodong Dou, Lan Jiang, Hongwei Jin, Lihe Zhang, Liangren Zhang*, Zhenming Liu*. Discovery of novel glycogen synthase kinase-3 alpha inhibitors: Structure-based virtual screening, preliminary SAR and biological evaluation for treatment of acute myeloid leukemia. Eur J Med Chem., 2019, 171, 221-234.
  30. Lixin Yang, Ting Li, Songlu Li, Yang Wu, Xiaomeng Shi, Hongwei Jin, Zhenming Liu, Yongjuan Zhao*, Liangren Zhang*, Hon Cheung Lee, Lihe Zhang. Rational Design and Identification of Small-Molecule Allosteric Inhibitors of CD38. ChemBioChem, 2019, 20(19), 2485-2493.
  31. Lixin Yang, Yongqing Liu, Minghua Fan, Guiwang Zhu, Hongwei Jin, Jing Liang, Zhenming Liu, Zhuo Huang*, Liangren Zhang*. Identi？cation and characterization of benzo[d]oxazol-2(3H)-one derivatives as the first potent and selective small-molecule inhibitors of chromodomain protein CDYL. Eur. J. Med. Chem., 2019, 182, 111656.

 

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